Kinetic and Spatial Analysis of Intracellular Signal Transduction Networks

 

Jason Haugh

Department of Chemical and Biomolecular Engineering

North Carolina State University

 

An ongoing challenge in mammalian cell biology is to bridge the gaps in our understanding of processes at the molecular, cellular, and tissue levels.  Central to the hierarchy of biological complexity is the field of signal transduction, which deals with the biochemical mechanisms and pathways by which cells respond to external stimuli, such as soluble growth factors/cytokines, immobilized ligands such as those found in extracellular matrix or the surfaces of other cells, and mechanical forces.  Intracellular signaling processes control the growth, survival, and migration of cells in normal physiological contexts, and defects in signaling form the molecular basis for cancer, immune system disorders, and other diseases.  Using a quantitative approach that combines biochemical measurements, live-cell fluorescence microscopy, and mathematical modeling, we seek to characterize signal transduction networks through analysis of their kinetics and spatial patterns in cells.  Based on analysis of experimental data and informed where appropriate by knowledge of protein domain structure, mechanistic models are developed that may be embedded (in coarse-grained form) in mathematical representations of cell population dynamics, with the goal of evaluating hypotheses regarding the concerted responses of cells in tissues.

 

As an example of this approach, our efforts to characterize signal transduction mediated by cell surface receptors for platelet-derived growth factor (PDGF), a soluble factor that accelerates dermal wound healing by directing the migration and proliferation of dermal fibroblasts, will be described in two parts.  In the first part of the talk, I will describe spatial modeling and subcellular characterization of the signaling mechanism by which fibroblasts sense PDGF gradients, which in turn has led us to analyze tissue-scale models of wound invasion driven by such gradients.  The second part of the talk will cover the elucidation and kinetic characterization of the so-called crosstalk interactions between two canonical signaling pathways strongly activated by PDGF receptors (Ras/Erk and PI 3-kinase), which has moved us towards predictive modeling at the level of signal transduction networks.